2020

  • Rational design, synthesis and biological profiling of new KDM4C inhibitorsBioorg. Med. Chem. 2020, 28, 115128
  • Pharmacokinetic Evaluation of Brain Penetrating Morpholine-3-hydroxy-2-pyridine Oxime as an Antidote for Nerve Agent Poisoning ACS Chem. Neurosci. 2020, 11, 7, 1072-1084
  • Growth, health aspects and histopathology of brown bullhead (Ameiurus nebulosus L.): replacing fishmeal with soybean meal and brewer’s yeast

Scientific Reports. 2020, 10, 1104

  • Clarithromycin inhibits autophagy in colorectal cancer by regulating the hERG1 potassium channel interaction with                                                                                          PI3K Cell Death Dis. 11, 161, 2020 

2019

  • Pro-inflammatory effects of extracellular Hsp70 on NCI-H292 human bronchial epithelial cell line                                                                                                                        Int. J. Clin. Exp. Pathol. 2019, 100, 320-329
  • Preventing lung pathology and mortality in rabbit Staphylococcus aureus pneumonia models with cytotoxin-neutralizing monoclonal IgGs penetrating the epithelial lining fluid Scientific Reports, 2019, 9, 5339 
  • Precision-cut lung slices from bleomycin treated animals as a model for testing potential therapies for idiopathic pulmonary fibrosis                                                              Pulm. Pharmacol. Ther. 2019, 55, 75-83  
  • Macrolides: Properties, Synthesis and Applications                                                                                                                                                                        ChemMedChem, 2019, 14, 359
  • Lipophilicity and bio-mimetic properties determination of phytoestrogens using ultra-high-performance liquid chromatography
  • Biomedical Chromatography, 2019, 33:e4551
  • Effects of extracellular Hsp70 and cigarette smoke on differentiated THP-1 cells and human monocyte-derived macrophages                                                                           Mol. Immunol. 2019, 111, 53-63
  • Comparative study of polyphenolic composition and anti-inflammatory activity of Thymus species                                                                                                                 Eur. Food Res. Technol. 245, 2019, 1951–1962
  • Benzoxaboroles-novel autotaxin inhibitors                                                                                                                                                                                           Molecules, 2019, 24, 3419
  • Association of NLRP1 Coding Polymorphism with Lung Function and Serum IL-1β Concentration in Patients Diagnosed with Chronic Obstructive Pulmonary Disease (COPD) Genes, 2019, 10, 783
  • Antiinflammatory and antiproliferative activity of naphthoxazole, fused hetero-benzoxazole and bridged benzobicyclic photoproducts                                                           Croatica Chemica Acta, 2019, 92, 191-201
  • Aflatoxin production and in vitro toxicity of Aspergilli section Flavi isolated from air samples collected from different environments                                                          Mycotoxin Res. 2019, 35, 217-230
  • A new screening tool to determine chameleonic properties of macrocycles                                                                                                                                                     J. Mol. Struct. 2019, 1198, 126929

2018

  • Small molecule purine and pseudopurine derivatives: synthesis, cytostatic evaluations and investigation of growth inhibitory effect in non-small cell lung cancer A549                   J. Enzyme Inhib. Med. Chem. 2018, 33:1, 271-285
  • Induction of Amyloid-β42 Production by Fipronil and Other Pyrazole Insecticides                                                                                                                                            J. Alzheimer’s Dis. 2018, vol. 62, no. 4, 1663-1681
  • Fumonisin production and toxic capacity in airborne black Aspergilli                                                                                                                                                         Toxicol In Vitro, 2018, vol. 53, 161-170
  • Extracellular Hsp70 induces inflammation and modulates LPS/LTA-stimulated inflammatory response in THP-1 cells                                                                                          Cell Stress Chaperones 2018, 23, 373-384 
  • Discovery of N-(3-Carbamoyl-5,5,7,7-tetramethyl-5,7-dihydro-4H-thieno[2,3-c]pyran-2-yl)-lH-pyrazole-5-carboxamide (GLPG1837), a Novel Potentiator Which Can Open Class III Mutant Cystic Fibrosis Transmembrane Conductance Regulator (CFTR) Channels to a High Extent                                                                                                                 J. Med. Chem. 2018, 61, 4, 1425-1435
  • Design, synthesis and biological evaluation of novel benzimidazole amidines as potent multi-target inhibitors for the treatment of non-small cell lung cancer                                Eur. J. Med. Chem. 2018, 143, 1616-1634  
  • Current Trends in Macrocyclic Drug Discovery and beyond-Ro5                                                                                                                                                                     Progress in Medicinal Chemistry, 2018, 57, 113-233
  • An alternative synthesis of the non-small cell lung carcinoma drug afatinib                                                                                                                                              Tetrahedron Letters, 2018, 59, 4180-4182
  • 16-membered macrolide antibiotics: a review                                                                                                                                                                                                 Int. J. Antimicrob. Agents, 2018, 51, 283-298

2017

  • Major Antimicrobial Representatives from Marine Sponges and/or Their Associated Bacteria                                                                                                                          Blue Biotechnology. Progress in Molecular and Subcellular Biology, vol 55. Springer, Cham
  • Discovery of 2-[[2-Ethyl-6-[4-[2-(3-hydroxyazetidin-1-yl)-2-oxoethyl]piperazin-1-yl]-8-methylimidazo[1,2-a]pyridin-3-yl]methylamino]-4-(4-fluorophenyl)thiazole-5-carbonitrile (GLPG1690), a First-in-Class Autotaxin Inhibitor Undergoing Clinical Evaluation for the Treatment of Idiopathic Pulmonary Fibrosis                                                                 Eur. J.Med. Chem. 2017, 60, 9, 3580-3590
  • Discovery and Development of Novel Drugs                                                                                                                                                                                               Blue Biotechnology. Progress in Molecular and Subcellular Biology, vol 55. Springer, Cham
  • Comparison of antitumor activity of some benzothiophene and thienothiophene carboxanilides and quinolones in 2D and 3D cell culture system                                                   Croat. Chem. Acta 2017, 90(3), 413–424
  • Around the macrolide – Impact of 3D structure of macrocycles on lipophilicity and cellular accumulation.                                                                                                        Eur. J. Med. Chem. 2017, 133, 351-364
  • Antiproliferative activity of amino substituted benzo[b]thieno[2,3-b]pyrido[1,2-a]benzimidazoles explored by 2D and 3D cell culture system                                                           Eur. J. Med. Chem. 2017, 125, 722-735

2016

  • Reinvestigation of the Branimycin Stereochemistry at Position 17-C                                                                                                                                                             Org. Lett. 2016, 18, 4, 780-783 
  • Macrolones Are a Novel Class of Macrolide Antibiotics Active against Key Resistant Respiratory Pathogens In Vitro and In Vivo                                                                       Antimicrobial Agents and Chemotherapy Aug 2016, 60 (9) 5337-5348
  • From erythromycin to azithromycin and new potential ribosome-binding antimicrobials                                                                                                                                   Antibiotics 2016, 5(3), 29
  • Baicalin and baicalein inhibit Src tyrosine kinase and production of IL-6                                                                                                                                                          J Chem, Vol 2016, 2510621/1-2510621/6
  • Antitumor activity of amidino-substituted benzimidazole and benzimidazo[1,2-a]quinoline derivatives tested in 2D and 3D cell culture systems                                                  Journal of Enzyme Inhibition and Medicinal Chemistry, 31:6, 1139-1145
  • A comprehensive evaluation of novel oximes in creation of butyrylcholinesterase-based nerve agent bioscavengers                                                                                   Toxicol. Appl. Pharmacol. 2016, 310, 195-204

2015

  • Structure and conformational analysis of spiroketals from 6-O-methyl-9(E)-hydroxyiminoerythronolide A                                                                                                Beilstein J. Org. Chem. 2015, 11, 1447–1457
  • Relative potencies of three glucocorticoids to induce hypoplasia of the physis and concomitant biochemical alterations in the rat                                                                      Drug and Chemical Toxicology, 38:3, 272-277
  • Ethers from esters; from exceptional transformationto synthetic method                                                                                                                                                Arkivoc, Vol 2015, Issue 1, Reviews and Accounts, 300-326 
  • Bacterial DNA gyrase and topoisomerase IV are essential enzymes that control the topological state of DNA during replication and validated antibacterial drug targets                  J. Med. Chem. 2015, 58, 14, 5501-5521 

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